One-Pot Double Cyclizations Involving an Aza-Prins Process
Overview & Synopsis
Piperidine derivatives are highly abundant in natural products and pharmaceutically relevant compounds. Aza-Prins cyclization has emerged as a step-atom-economical and stereoselective method for the preparation of such azacycles. The possibility of coupling aza-Prins process with the formation of a second cycle in a one-pot manner is even more powerful and makes the object of this review. Cascade/domino/tandem bis-cyclizations involving an aza-Prins process, for the rapid construction of complex small molecules, are discussed in detail.Scheme 7. Tandem cyclisation towards azasteroids.
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Document Information
| Document Title | One-Pot Double Cyclizations Involving an Aza-Prins Process |
|---|---|
| Author / Organization | Nicolas Gouault, Maxence Roydor, Jacques Renault, Swarnayu Banik, B V Subba Reddy, Claudia Lalli |
| Subject & Discipline | Multidisciplinary Academic Open Research |
| Categories | Science & Mathematics |
| Publication Year | 2024 |
| License / Rights | Open Access / Creative Commons |
| Resource Verification | Listed PDF (Verification Pending) |
| Original Host Website |
HAL Open Science
(hal.science)
|
| File Format | application/pdf (Portable Document Format) |
| Language | EN |
| Catalog ID | DOC-107651 |
| Original Source Link | Visit Source Page on hal.science » |